Publications
2020
Valero T., Baillache D.J., Fraser C., Myers S.H., Unciti-Broceta A.
Pyrazolopyrimide library screening in glioma cells discovers highly potent antiproliferative leads that target the PI3K/mTOR pathway
Bioorganic and Medicinal Chemistry, vol. 28, (no. 1)
2020
Myers S.H., Ortega J.A., Cavalli A.
Synthetic Lethality through the Lens of Medicinal Chemistry
Journal of Medicinal Chemistry, vol. 63, (no. 23), pp. 14151-14183
2019
Conole D., Myers S.H., Mota F., Hobbs A.J., Selwood D.L.
Biophysical screening methods for extracellular domain peptide receptors, application to natriuretic peptide receptor C ligands
Chemical Biology and Drug Design, vol. 93, (no. 6), pp. 1011-1020
2019
Cruz-Lopez O., Temps C., Longo B., Myers S.H., Franco-Montalban F., Unciti-Broceta A.
Synthesis and Characterization of a Click-Assembled 18-Atom Macrocycle That Displays Selective AXL Kinase Inhibitory Activity
ACS Omega, vol. 4, (no. 25), pp. 21620-21626
2018
Myers S.H., Temps C., Houston D.R., Brunton V.G., Unciti-Broceta A.
Development of Potent Inhibitors of Receptor Tyrosine Kinases by Ligand-Based Drug Design and Target-Biased Phenotypic Screening
Journal of Medicinal Chemistry, vol. 61, (no. 5), pp. 2104-2110
2016
Myers S.H., Brunton V.G., Unciti-Broceta A.
AXL Inhibitors in Cancer: A Medicinal Chemistry Perspective
Journal of Medicinal Chemistry, vol. 59, (no. 8), pp. 3593-3608
2014
Weiss J.T., Fraser C., Rubio-Ruiz B., Myers S.H., Crispin R., Dawson J.C., Brunton V.G., Patton E.E., Carragher N.O., Unciti-Broceta A.
N-alkynyl derivatives of 5-fluorouracil: Susceptibility to palladium-mediated dealkylation and toxigenicity in cancer cell culture
Frontiers in Chemistry, vol. 2, (no. JUL)