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People ■ Giampiero Colombano
Giampiero Colombano's foto

Giampiero Colombano

Post Doc

iit / Drug Discovery and Development


Phone +39 010 71781921

Selected Publications

1. Appendino G., Prosperini S., Valdivia C., Ballero M., Colombano G., Billington R.A., Genazzani A.A., Sterner O. "SERCA-inhibiting activity of C-19 Terpenolides from Thapsia garganica and their possible biogenesis". Journal of Natural Products 2005, 68, 1213-7.

2. Colombano G., Travelli C., Galli U., Caldarelli A., Chini M.G., Canonico P.G., Sorba G., Bifulco G., Tron G.C., and Genazzani A.A. "A novel potent nicotinamide phosphoribosyltransferase inhibitor synthesized via click chemistry". J. Med. Chem. 2010, 53 (2), 616-623.

3. Mossetti R., Caprioglio D., Colombano G., Tron G.C., Pirali T. "A novel a-isocyanoacetamide-based three-component reaction for the synthesis of dialkyl 2-acyl-5-aminofuran-3,4-dicarboxylates". Org. Biomol. Chem., 2011, 9, 1627-1631.

4. Sasso O., Bertorelli R., Bandiera T., Scarpelli R., Colombano G., Armirotti A., Moreno-Sanz G., Reggiani A., Piomelli D. "Peripheral FAAH inhibition causes profund antinociception and proptects against indomethacin-induced gastric lesions". Pharmacol Res.,2012, 65, 553-563.

5. Bassetto, M., De Burghgraeve, T., Delang, L., Massarotti, A., Coluccia, A., Zonta, N., Gatti, V., Colombano, G., Sorba, G., Silvestri, R., Tron, G.C., Neyts, J., Leyssen, P., Brancale, A. "Computer-aided identification, design and synthesis of a novel series of compounds with selective antiviral activity against chikungunya virus". Antiviral Research, 2013, 98, 12-18.

 

 

1. Appendino G., Prosperini S., Valdivia C., Ballero M., Colombano G., Billington R.A., Genazzani A.A., Sterner O. "SERCA-inhibiting activity of C-19 Terpenolides from Thapsia garganica and their possible biogenesis". Journal of Natural Products 2005, 68, 1213-7.

2. Colombano G., Travelli C., Galli U., Caldarelli A., Chini M.G., Canonico P.G., Sorba G., Bifulco G., Tron G.C., and Genazzani A.A. "A novel potent nicotinamide phosphoribosyltransferase inhibitor synthesized via click chemistry". J. Med. ...

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